PRE-084 hydrochloride boxaldehyde 6 nM in a FLAP

6 nM in a FLAP binding assay

Chemical Name: Compound Library of Histone Demethylase

TBK1/IKKε-IN-1(compound 1) effectively blocks immune suppressive cytokine elaboration by CT26 cell line spheroids

Thiamet-G is a potent inhibitor of the enzyme O-GlcNAcase (Ki = 21 nM)

PRE-084 hydrochloride boxaldehyde 6 nM in a FLAPPRE 084 hydrochloride is a high affinity, selective 1 agonist, has an IC50 of 44 nM in the sigma receptor assay. IC50 value: 44 nMTarget: sigma receptorin vitro: PRE 084 has an IC50 of more than 100,000 nM for PCP receptors and an IC50 higher than 10,000 nM in a variety of other receptor systems. in vivo: PRE 084 improves motor neuron survival and motor performance in wobbler mice. PRE 084 enhances BDNF mediated trophic support. Product information